Posted by Skeletor on November 17, 2020, at 15:11:08
In reply to Re: 5HT2 antagonist without anticholinergic properties » jay2112, posted by Skeletor on November 17, 2020, at 15:07:41
This is kinda interesting: https://en.wikipedia.org/wiki/Deramciclane
---------------------------------------------------------------------------What is your take on Amoxapine?
https://en.wikipedia.org/wiki/Amoxapine
---------------------------------------------------------------------------For Pizotifen I get the following values from Ki Database https://en.wikipedia.org/wiki/Pizotifen
5HT1A... 200 - 1700 nM
5HT2A... 15.5 nM
5HT2C... 5 - 8 nM
I didn't find values for H1 and muscarinic receptors
---------------------------------------------------------------------------https://en.wikipedia.org/wiki/Ritanserin
Also quite strong at 5HT2
Then there is also stuff like Ketanserin, Pimavanserin etc.
---------------------------------------------------------------------------https://en.wikipedia.org/wiki/Nefazodone
Pretty perfect drug ^^
Never understood its ban.
poster:Skeletor
thread:1112581
URL: http://www.dr-bob.org/babble/20201025/msgs/1112597.html